PDB entry 4r5s
View 4r5s on RCSB PDB site
Description: Crystal structure of EGFR 696-1022 L858R in complex with FIIN-3
Class: transferase
Keywords: EGFR, L858R, Kinase, FIIN-3, TRANSFERASE
Deposited on
2014-08-22, released
2014-11-12
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-11-12, with a file datestamp of
2014-11-07.
Experiment type: XRAY
Resolution: 3 Å
R-factor: 0.203
AEROSPACI score: 0.18
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
- Uniprot P00533
- engineered mutation (166)
Domains in SCOPe 2.08: d4r5sa_ - Heterogens: FI3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4r5sA (A:)
gspsgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreat
spkankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigs
qyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakllgaeekeyha
eggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekge
rlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlps
ptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>4r5sA (A:)
eapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatspkan
keildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqylln
wcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakllgaeevpikwmales
ilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvym
imvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpedmddvvdadeyli