PDB entry 4qp9
View 4qp9 on RCSB PDB site
Description: Crystal Structure of ERK2 in complex with 7-(1-propyl-1H-pyrazol-4-yl)-2-(pyridin-4-yl)-5H-pyrrolo[2,3-b]pyrazine
Class: transferase/transferase inhibitor
Keywords: Kinase, transferase-transferase inhibitor complex
Deposited on
2014-06-22, released
2015-09-23
The last revision prior to the SCOPe 2.08 freeze date was dated
2015-12-16, with a file datestamp of
2015-12-11.
Experiment type: XRAY
Resolution: 2 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAPK1, ERK2, PRKM1, PRKM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4qp9a_ - Heterogens: 35X, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4qp9A (A:)
mgshhhhhhmaaaaaagagpemvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrv
aikkispfehqtycqrtlreikillrfrheniigindiiraptieqmkdvyivqdlmetd
lykllktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfgla
rvadpdhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgk
hyldqlnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfpnadskaldlld
kmltfnphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeet
arfqpgyrs
Sequence, based on observed residues (ATOM records): (download)
>4qp9A (A:)
mvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrvaikkispfehqtycqrtlrei
killrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyflyq
ilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadlteyvatrwyrapeiml
nskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqedlnciinlka
rnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalahpyleqyydps
depiaeapfkfelddlpkeklkelifeetarfqpg