PDB entry 4qm0
View 4qm0 on RCSB PDB site
Description: Crystal structure of RORc in complex with a tertiary sulfonamide inverse agonist
Class: Transcription/Transcription inhibitor
Keywords: nuclear receptor ligand binding domain, Transcription-Transcription inhibitor complex
Deposited on
2014-06-14, released
2014-09-17
The last revision prior to the SCOPe 2.06 freeze date was dated
2014-09-17, with a file datestamp of
2014-09-12.
Experiment type: XRAY
Resolution: 2.19 Å
R-factor: 0.186
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Nuclear receptor ROR-gamma
Species: Homo sapiens [TaxId:9606]
Gene: RORC, NR1F3, RORG, RZRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4qm0a_ - Chain 'C':
Compound: Nuclear receptor ROR-gamma
Species: Homo sapiens [TaxId:9606]
Gene: RORC, NR1F3, RORG, RZRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4qm0c1, d4qm0c2 - Heterogens: 39K, DMS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4qm0A (A:)
gsapyaslteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwer
cahhlteaiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffe
gkyggmelfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkv
eqlqynlelafhhhlckthrqsilaklppkgklrslcsqhverlqifqhlhpivvqaafp
plykelfsgns
Sequence, based on observed residues (ATOM records): (download)
>4qm0A (A:)
aslteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwercahhl
teaiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffegkygg
melfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkveqlqy
nlelafhhhlckthrqsilaklppkgklrslcsqhverlqifqhlhpivvqaaf
- Chain 'C':
Sequence, based on SEQRES records: (download)
>4qm0C (C:)
gsapyaslteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwer
cahhlteaiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffe
gkyggmelfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkv
eqlqynlelafhhhlckthrqsilaklppkgklrslcsqhverlqifqhlhpivvqaafp
plykelfsgns
Sequence, based on observed residues (ATOM records): (download)
>4qm0C (C:)
aslteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwercahhl
teaiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffegkygg
melfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkveqlqy
nlelafhhhlckthrqsilaklppkgklrslcsqhverlqqaafpplykelfsgns