PDB entry 4nvq
View 4nvq on RCSB PDB site
Description: Human G9a in Complex with Inhibitor A-366
Class: Transferase/Transferase Inhibitor
Keywords: Lysine Methyl Transferase, Transferase-Transferase Inhibitor complex
Deposited on
2013-12-05, released
2014-01-15
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-22, with a file datestamp of
2017-11-17.
Experiment type: XRAY
Resolution: 2.03 Å
R-factor: N/A
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Histone-lysine N-methyltransferase EHMT2
Species: Homo sapiens [TaxId:9606]
Gene: EHMT2, BAT8, C6orf30, G9A, KMT1C, NG36
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4nvqa_ - Chain 'B':
Compound: Histone-lysine N-methyltransferase EHMT2
Species: Homo sapiens [TaxId:9606]
Gene: EHMT2, BAT8, C6orf30, G9A, KMT1C, NG36
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4nvqb_ - Heterogens: 2OD, SAH, ZN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4nvqA (A:)
gshmnrairtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrni
thlqhctcvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrnck
nrvvqsgikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfd
ldnkdgevycidaryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtge
elgfdygdrfwdikskyftcqcgsekckhsaeaialeqsrlarld
Sequence, based on observed residues (ATOM records): (download)
>4nvqA (A:)
irtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrnithlqhct
cvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrncknrvvqsg
ikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfdlgevyci
daryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtgeelgfdygdrfw
diksyftcqcgsekckhsaeaialeqs
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4nvqB (B:)
gshmnrairtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrni
thlqhctcvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrnck
nrvvqsgikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfd
ldnkdgevycidaryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtge
elgfdygdrfwdikskyftcqcgsekckhsaeaialeqsrlarld
Sequence, based on observed residues (ATOM records): (download)
>4nvqB (B:)
tekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrnithlqhctcv
ddcsssnclcrcwydkdgrllqefnkiepplifecnqacscwrncknrvvqsgikvrlql
yrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfdldvycidaryygni
srfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtgeelgfdygdrfwdikskyft
cqcgsekckhsaeaialeqsrla