PDB entry 4nvq

View 4nvq on RCSB PDB site
Description: Human G9a in Complex with Inhibitor A-366
Class: Transferase/Transferase Inhibitor
Keywords: Lysine Methyl Transferase, Transferase-Transferase Inhibitor complex
Deposited on 2013-12-05, released 2014-01-15
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-11-22, with a file datestamp of 2017-11-17.
Experiment type: XRAY
Resolution: 2.03 Å
R-factor: N/A
AEROSPACI score: 0.3 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Histone-lysine N-methyltransferase EHMT2
    Species: Homo sapiens [TaxId:9606]
    Gene: EHMT2, BAT8, C6orf30, G9A, KMT1C, NG36
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4nvqa_
  • Chain 'B':
    Compound: Histone-lysine N-methyltransferase EHMT2
    Species: Homo sapiens [TaxId:9606]
    Gene: EHMT2, BAT8, C6orf30, G9A, KMT1C, NG36
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4nvqb_
  • Heterogens: 2OD, SAH, ZN, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4nvqA (A:)
    gshmnrairtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrni
    thlqhctcvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrnck
    nrvvqsgikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfd
    ldnkdgevycidaryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtge
    elgfdygdrfwdikskyftcqcgsekckhsaeaialeqsrlarld
    

    Sequence, based on observed residues (ATOM records): (download)
    >4nvqA (A:)
    irtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrnithlqhct
    cvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrncknrvvqsg
    ikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfdlgevyci
    daryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtgeelgfdygdrfw
    diksyftcqcgsekckhsaeaialeqs
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >4nvqB (B:)
    gshmnrairtekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrni
    thlqhctcvddcsssnclcgqlsircwydkdgrllqefnkiepplifecnqacscwrnck
    nrvvqsgikvrlqlyrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfd
    ldnkdgevycidaryygnisrfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtge
    elgfdygdrfwdikskyftcqcgsekckhsaeaialeqsrlarld
    

    Sequence, based on observed residues (ATOM records): (download)
    >4nvqB (B:)
    tekiicrdvargyenvpipcvngvdgepcpedykyisencetstmnidrnithlqhctcv
    ddcsssnclcrcwydkdgrllqefnkiepplifecnqacscwrncknrvvqsgikvrlql
    yrtakmgwgvralqtipqgtficeyvgelisdaeadvreddsylfdldvycidaryygni
    srfinhlcdpniipvrvfmlhqdlrfpriaffssrdirtgeelgfdygdrfwdikskyft
    cqcgsekckhsaeaialeqsrla