PDB entry 4npv
View 4npv on RCSB PDB site
Description: Crystal structure of human PDE1B bound to inhibitor 7A (6,7,8-trimethoxy-N-(pentan-3-yl)quinazolin-4-amine)
Class: hydrolase/hydrolase inhibitor
Keywords: HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2013-11-22, released
2014-07-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-07-16, with a file datestamp of
2014-07-11.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.207
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
Species: Homo sapiens [TaxId:9606]
Gene: PDE1B, PDE1B1, PDES1B
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4npva_ - Heterogens: 0NK, MG, ZN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4npvA (A:)
gsmtytsvgptystavlnclknldlwcfdvfslnqaaddhalrtivfelltrhnlisrfk
iptvflmsfldaletgygkyknpyhnqihaadvtqtvhcfllrtgmvhclseiellaiif
aaaihdyehtgttnsfhiqtksecaivyndrsvlenhhissvfrlmqddemnifinltkd
efvelralviemvlatdmschfqqvktmktalqqleridkpkalslllhaadishptkqw
lvhsrwtkalmeeffrqgdkeaelglpfsplcdrtstlvaqsqigfidfiveptfsvltd
vaeksvqpladedsksknqpsfqwrqpsldvevgdpnpdvvsfrstwvkriqenkqkwke
raasgitnq
Sequence, based on observed residues (ATOM records): (download)
>4npvA (A:)
stavlnclknldlwcfdvfslnqaaddhalrtivfelltrhnlisrfkiptvflmsflda
letgygkyknpyhnqihaadvtqtvhcfllrtgmvhclseiellaiifaaaihdyehtgt
tnsfhiqtksecaivyndrsvlenhhissvfrlmqddemnifinltkdefvelralviem
vlatdmschfqqvktmktalqqleridkpkalslllhaadishptkqwlvhsrwtkalme
effrqgdkeaelglpfsplcdrtstlvaqsqigfidfiveptfsvltdvaeksvqppdvv
sfrstwvkriqenkqkwkeraas