PDB entry 4nka
View 4nka on RCSB PDB site
Description: Crystal structure of human fibroblast growth factor receptor 1 kinase domain in complex with pyrazolaminopyrimidine 2
Class: transferase/transferase inhibitor
Keywords: KINASE, ATP BINDING, PHOSPHORYLATION, TRANS-MEMBRANE, transferase-transferase inhibitor complex
Deposited on
2013-11-12, released
2013-12-18
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-07-16, with a file datestamp of
2014-07-11.
Experiment type: XRAY
Resolution: 2.19 Å
R-factor: 0.2
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4nkaa_ - Chain 'B':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4nkab_ - Heterogens: SO4, EDO, 2K7, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4nkaA (A:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>4nkaA (A:)
elpedprwelprdrlvlgkplgeqvvlaeaigldkdkpnrvtkvavkmlksdatekdlsd
lisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppeeqlsskd
lvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfgidyykkttngrlpvkw
mapealfdriythqsdvwsfgvllweiftlggspypgvpveelfkllkeghrmdkpsnct
nelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4nkaB (B:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>4nkaB (B:)
agvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkpnrvtkvavkmlksd
atekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrpp
eqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfhhidyykktt
ngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelfkllkeghr
mdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe