PDB entry 4myq
View 4myq on RCSB PDB site
Description: Selective Inhibition of the Catalytic Domain Of Human Phosphodiesterase 4B With A-33
Class: hydrolase/hydrolase inhibitor
Keywords: PHOSPHODIESTERASE, CATALYTIC, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2013-09-27, released
2014-01-01
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-15, with a file datestamp of
2017-11-10.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: N/A
AEROSPACI score: 0.35
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP-specific 3',5'-cyclic phosphodiesterase 4B
Species: Homo sapiens [TaxId:9606]
Gene: DPDE4, PDE4, PDE4B
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4myqa_ - Heterogens: 19T, MG, ZN, NA, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4myqA (A:)
gshmsisrfgvntenedhlakeledlnkwglnifnvagyshnrpltcimyaifqerdllk
tfrissdtfitymmtledhyhsdvayhnslhaadvaqsthvllstpaldavftdleilaa
ifaaaihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqeehcdifmnlt
kkqrqtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvllldnytdriqvlrnm
vhcadlsnptkslelyrqwtdrimeeffqqgdkerergmeispmcdkhtasveksqvgfi
dyivhplwetwadlvqpdaqdildtlednrnwyqsmipqspsppldeqnrdcqglmekfq
feltldeedseg
Sequence, based on observed residues (ATOM records): (download)
>4myqA (A:)
sisrfgvntenedhlakeledlnkwglnifnvagyshnrpltcimyaifqerdllktfri
ssdtfitymmtledhyhsdvayhnslhaadvaqsthvllstpaldavftdleilaaifaa
aihdvdhpgvsnqflintnselalmyndesvlenhhlavgfkllqeehcdifmnltkkqr
qtlrkmvidmvlatdmskhmslladlktmvetkkvtssgvllldnytdriqvlrnmvhca
dlsnptkslelyrqwtdrimeeffqqgdkerergmeispmcdkhtasveksqvgfidyiv
hplwetwadlvqpdaqdildtlednrnwyqsmipqcqglmekfqf