PDB entry 4luc
View 4luc on RCSB PDB site
Description: Crystal Structure of small molecule disulfide 6 bound to K-Ras G12C
Class: signaling protein/inhibitor
Keywords: GTPase, GDP bound, SIGNALING PROTEIN-INHIBITOR complex
Deposited on
2013-07-25, released
2013-11-27
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-12-18, with a file datestamp of
2013-12-13.
Experiment type: XRAY
Resolution: 1.29 Å
R-factor: 0.152
AEROSPACI score: 0.69
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS isoform 2B, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
- Uniprot P01116 (1-End)
- variant (12)
- engineered mutation (51)
- engineered mutation (80)
- engineered mutation (118)
- see remark 999 (151)
- see remark 999 (153)
- see remark 999 (165-168)
Domains in SCOPe 2.05: d4luca_ - Chain 'B':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS isoform 2B, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
- Uniprot P01116 (1-End)
- variant (12)
- engineered mutation (51)
- engineered mutation (80)
- engineered mutation (118)
- see remark 999 (151)
- see remark 999 (153)
- see remark 999 (165-168)
Domains in SCOPe 2.05: d4lucb_ - Heterogens: CA, 20G, GDP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4lucA (A:)
gmteyklvvvgacgvgksaltiqliqnhfvdeydptiedsyrkqvvidgetslldildta
gqeeysamrdqymrtgegfllvfainntksfedihhyreqikrvkdsedvpmvlvgnksd
lpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhkek
Sequence, based on observed residues (ATOM records): (download)
>4lucA (A:)
mteyklvvvgacgvgksaltiqliqnhfvdeydptiedsyrkqvvidgetslldildtag
qeeysamrdqymrtgegfllvfainntksfedihhyreqikrvkdsedvpmvlvgnksdl
psrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhke
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4lucB (B:)
gmteyklvvvgacgvgksaltiqliqnhfvdeydptiedsyrkqvvidgetslldildta
gqeeysamrdqymrtgegfllvfainntksfedihhyreqikrvkdsedvpmvlvgnksd
lpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhkek
Sequence, based on observed residues (ATOM records): (download)
>4lucB (B:)
mteyklvvvgacgvgksaltiqliqnhfvdeydptiedsyrkqvvidgetslldildtag
qeeysamrdqymrtgegfllvfainntksfedihhyreqikrvkdsedvpmvlvgnksdl
psrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhke