PDB entry 4kab
View 4kab on RCSB PDB site
Description: FOCAL ADHESION KINASE CATALYTIC DOMAIN IN COMPLEX WITH 3-Methyl-1,4-dihydro-pyrazolo[4,5-c]pyrazole
Class: Transferase/Transferase Inhibitor
Keywords: TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, Transferase-Transferase Inhibitor complex
Deposited on
2013-04-22, released
2013-09-11
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-10-09, with a file datestamp of
2013-10-04.
Experiment type: XRAY
Resolution: 2.71 Å
R-factor: 0.173
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Focal adhesion kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: PTK2, FAK, FAK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4kaba_ - Chain 'B':
Compound: Focal adhesion kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: PTK2, FAK, FAK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4kabb_ - Heterogens: 4KA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4kabA (A:)
gspstrdyeiqrerielgrcigegqfgdvhqgiymspenpalavaiktcknctsdsvrek
flqealtmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilya
yqlstalayleskrfvhrdiaarnvlvssndcvklgdfglsrymedstyykaskgklpik
wmapesinfrrftsasdvwmfgvcmweilmhgvkpfqgvknndvigriengerlpmppnc
pptlyslmtkcwaydpsrrprftelkaqlstileeekaq
Sequence, based on observed residues (ATOM records): (download)
>4kabA (A:)
trdyeiqrerielgrcigegqfgdvhqgiymsppalavaiktcknctsdsvrekflqeal
tmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilyayqlsta
layleskrfvhrdiaarnvlvssndcvklgdflpikwmapesinfrrftsasdvwmfgvc
mweilmhgvkpfqgvknndvigriengerlpmppncpptlyslmtkcwaydpsrrprfte
lkaqlstileeekaq
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4kabB (B:)
gspstrdyeiqrerielgrcigegqfgdvhqgiymspenpalavaiktcknctsdsvrek
flqealtmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilya
yqlstalayleskrfvhrdiaarnvlvssndcvklgdfglsrymedstyykaskgklpik
wmapesinfrrftsasdvwmfgvcmweilmhgvkpfqgvknndvigriengerlpmppnc
pptlyslmtkcwaydpsrrprftelkaqlstileeekaq
Sequence, based on observed residues (ATOM records): (download)
>4kabB (B:)
dyeiqrerielgrcigegqfgdvhqgiymspepalavaiktcknctsdsvrekflqealt
mrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilyayqlstal
ayleskrfvhrdiaarnvlvssndcvklgdfglsrymlpikwmapesinfrrftsasdvw
mfgvcmweilmhgvkpfqgvknndvigriengerlpmppncpptlyslmtkcwaydpsrr
prftelkaqlstileeek