PDB entry 4k9y
View 4k9y on RCSB PDB site
Description: FOCAL ADHESION KINASE Catalytic domain in complex with 1-[4-(6-Amino-purin-9-yl)-phenyl]-3-(5-tert-butyl-2-p-tolyl-2H-pyrazol-3-yl)-urea
Class: Transferase/Transferase Inhibitor
Keywords: TYROSINE PROTEIN KINASE, TRANSFERASE, ATP BINDING, Transferase-Transferase Inhibitor complex
Deposited on
2013-04-21, released
2013-09-11
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-10-09, with a file datestamp of
2013-10-04.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.165
AEROSPACI score: 0.49
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Focal adhesion kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: PTK2, FAK, FAK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4k9ya_ - Heterogens: K9Y, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4k9yA (A:)
gspstrdyeiqrerielgrcigegqfgdvhqgiymspenpalavaiktcknctsdsvrek
flqealtmrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilya
yqlstalayleskrfvhrdiaarnvlvssndcvklgdfglsrymedstyykaskgklpik
wmapesinfrrftsasdvwmfgvcmweilmhgvkpfqgvknndvigriengerlpmppnc
pptlyslmtkcwaydpsrrprftelkaqlstileeekaq
Sequence, based on observed residues (ATOM records): (download)
>4k9yA (A:)
yeiqrerielgrcigegqfgdvhqgiymspenpalavaiktcknctsdsvrekflqealt
mrqfdhphivkligvitenpvwiimelctlgelrsflqvrkysldlaslilyayqlstal
ayleskrfvhrdiaarnvlvssndcvklgdfglsrymedstyykaskgklpikwmapesi
nfrrftsasdvwmfgvcmweilmhgvkpfqgvknndvigriengerlpmppncpptlysl
mtkcwaydpsrrprftelkaqlstileeeka