PDB entry 4k7a
View 4k7a on RCSB PDB site
Description: Crystal structure of the androgen receptor ligand binding domain in complex with minoxidil
Class: transcription
Keywords: Aandrogen receptor, ligand binding domain(LBD), steroid receptor coactivator, 5-alpha-dihydrotestosterone(DHT), prostate cancer, transcription factor, coactivator binding, cytosol, nucleas, TRANSCRIPTION
Deposited on
2013-04-16, released
2014-04-16
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-04-16, with a file datestamp of
2014-04-11.
Experiment type: XRAY
Resolution: 2.44 Å
R-factor: 0.192
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Androgen receptor
Species: Homo sapiens [TaxId:9606]
Gene: Ar
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4k7aa_ - Heterogens: DHT, MXD, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4k7aA (A:)
qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
vddqmaviqyswmglmvfamgwrsftnvnsamlyfapdlvfneyrmhksrmysqcvrmrh
lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknp
tscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsg
kvkpiyfht
Sequence, based on observed residues (ATOM records): (download)
>4k7aA (A:)
qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
vddqmaviqyswmglmvfamgwrsftnvnsamlyfapdlvfneyrmhksrmysqcvrmrh
lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiascsrrf
yqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsgkvkpiyf
ht