PDB entry 4k7a

View 4k7a on RCSB PDB site
Description: Crystal structure of the androgen receptor ligand binding domain in complex with minoxidil
Class: transcription
Keywords: Aandrogen receptor, ligand binding domain(LBD), steroid receptor coactivator, 5-alpha-dihydrotestosterone(DHT), prostate cancer, transcription factor, coactivator binding, cytosol, nucleas, TRANSCRIPTION
Deposited on 2013-04-16, released 2014-04-16
The last revision prior to the SCOPe 2.08 freeze date was dated 2014-04-16, with a file datestamp of 2014-04-11.
Experiment type: XRAY
Resolution: 2.44 Å
R-factor: 0.192
AEROSPACI score: 0.27 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Androgen receptor
    Species: Homo sapiens [TaxId:9606]
    Gene: Ar
    Database cross-references and differences (RAF-indexed):
    • Uniprot P10275 (0-248)
      • conflict (90)
    Domains in SCOPe 2.08: d4k7aa_
  • Heterogens: DHT, MXD, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4k7aA (A:)
    qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
    vddqmaviqyswmglmvfamgwrsftnvnsamlyfapdlvfneyrmhksrmysqcvrmrh
    lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiackrknp
    tscsrrfyqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsg
    kvkpiyfht
    

    Sequence, based on observed residues (ATOM records): (download)
    >4k7aA (A:)
    qpiflnvleaiepgvvcaghdnnqpdsfaallsslnelgerqlvhvvkwakalpgfrnlh
    vddqmaviqyswmglmvfamgwrsftnvnsamlyfapdlvfneyrmhksrmysqcvrmrh
    lsqefgwlqitpqeflcmkalllfsiipvdglknqkffdelrmnyikeldriiascsrrf
    yqltklldsvqpiarelhqftfdllikshmvsvdfpemmaeiisvqvpkilsgkvkpiyf
    ht