PDB entry 4jxv
View 4jxv on RCSB PDB site
Description: X-ray crystal structure of AmpC beta-lactamase from E. coli in complex with a non-covalent inhibitor 3-{[2-(4-CARBOXYPHENYL)ETHYL]SULFAMOYL}THIOPHENE-2-CARBOXYLIC ACID (compound 5)
Class: hydrolase/hydrolase inhibitor
Keywords: cephalosporinase, beta-lactamase, serine hydrolase, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2013-03-28, released
2014-04-30
The last revision prior to the SCOPe 2.04 freeze date was dated
2014-04-30, with a file datestamp of
2014-04-25.
Experiment type: XRAY
Resolution: 1.76 Å
R-factor: 0.199
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Beta-lactamase
Species: Escherichia coli [TaxId:83333]
Gene: ampC, ampA, b4150, JW4111
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4jxva_ - Chain 'B':
Compound: Beta-lactamase
Species: Escherichia coli [TaxId:83333]
Gene: ampC, ampA, b4150, JW4111
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4jxvb_ - Heterogens: 1MU, PO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>4jxvA (A:)
apqqindivhrtitplieqqkipgmavaviyqgkpyyftwgyadiakkqpvtqqtlfelg
svsktftgvlggdaiargeiklsdpttkywpeltakqwngitllhlatytagglplqvpd
evksssdllrfyqnwqpawapgtqrlyanssiglfgalavkpsglsfeqamqtrvfqplk
lnhtwinvppaeeknyawgyregkavhvspgaldaeaygvkstiedmarwvqsnlkpldi
nektlqqgiqlaqsrywqtgdmyqglgwemldwpvnpdsiingsdnkialaarpvkaitp
ptpavraswvhktgatggfgsyvafipekelgivmlanknypnparvdaawqilnalq
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>4jxvB (B:)
apqqindivhrtitplieqqkipgmavaviyqgkpyyftwgyadiakkqpvtqqtlfelg
svsktftgvlggdaiargeiklsdpttkywpeltakqwngitllhlatytagglplqvpd
evksssdllrfyqnwqpawapgtqrlyanssiglfgalavkpsglsfeqamqtrvfqplk
lnhtwinvppaeeknyawgyregkavhvspgaldaeaygvkstiedmarwvqsnlkpldi
nektlqqgiqlaqsrywqtgdmyqglgwemldwpvnpdsiingsdnkialaarpvkaitp
ptpavraswvhktgatggfgsyvafipekelgivmlanknypnparvdaawqilnalq