PDB entry 4i9z
View 4i9z on RCSB PDB site
Description: Crystal structure of the PDE5A1 catalytic domain in complex with novel inhibitors
Class: hydrolase/hydrolase inhibitor
Keywords: HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2012-12-05, released
2014-01-01
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-01-01, with a file datestamp of
2013-12-27.
Experiment type: XRAY
Resolution: 2.08 Å
R-factor: 0.202
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cGMP-specific 3',5'-cyclic phosphodiesterase
Species: Homo sapiens [TaxId:9606]
Gene: PDE5, PDE5A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4i9za_ - Heterogens: 5BA, ZN, MG, PEG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4i9zA (A:)
mgsshhhhhhssglvprgshmeetrelqslaaavvpsaqtlkitdfsfsdfelsdletal
ctirmftdlnlvqnfqmkhevlcrwilsvkknyrknvayhnwrhafntaqcmfaalkagk
iqnkltdleilalliaalshdldhrgvnnsyiqrsehplaqlychsimehhhfdqclmil
nspgnqilsglsieeykttlkiikqailatdlalyikrrgeffelirknqfnledphqke
lflamlmtacdlsaitkpwpiqqriaelvateffdqgdrerkelnieptdlmnrekknki
psmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalaeqq
Sequence, based on observed residues (ATOM records): (download)
>4i9zA (A:)
eetrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhev
lcrwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalshd
ldhrgvnnsylaqlychsimehhhfdqclmilnspgnqilsglsieeykttlkiikqail
atdlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpwpiqqriael
vateffdknkipsmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalae