PDB entry 4hyh
View 4hyh on RCSB PDB site
Description: X-RAY Crystal structure of compound 39 bound to human chk1 kinase domain
Class: transferase/transferase inhibitor
Keywords: SERINE/THREONINE-PROTEIN KINASE CHK1 INHIBITOR, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-11-13, released
2013-03-06
The last revision prior to the SCOPe 2.03 freeze date was dated
2013-05-01, with a file datestamp of
2013-04-26.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.204
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4hyha_ - Heterogens: 1AM, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4hyhA (A:)
mavpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicink
mlnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvy
lhgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellk
rrefhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsapla
llhkilvenpsaritipdikkdrwynkplkkgakrprvtsggvsespsg
Sequence, based on observed residues (ATOM records): (download)
>4hyhA (A:)
pfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkenikkeicinkmlnhenvvk
fyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithr
dikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepv
dvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilven
psaritipdikkdrwynkplkkg