PDB entry 4hnf

View 4hnf on RCSB PDB site
Description: Crystal structure of ck1d in complex with pf4800567
Class: transferase/transferase inhibitor
Keywords: ck1d, kinase, inhibitor, PF4800567, transferase-transferase inhibitor complex
Deposited on 2012-10-19, released 2012-11-14
The last revision prior to the SCOPe 2.03 freeze date was dated 2013-01-02, with a file datestamp of 2012-12-28.
Experiment type: XRAY
Resolution: 2.07 Å
R-factor: 0.241
AEROSPACI score: 0.37 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Casein kinase I isoform delta
    Species: Homo sapiens [TaxId:9606]
    Gene: CSNK1D, HCKID
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.03: d4hnfa_
  • Chain 'B':
    Compound: Casein kinase I isoform delta
    Species: Homo sapiens [TaxId:9606]
    Gene: CSNK1D, HCKID
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.03: d4hnfb_
  • Heterogens: 16W, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4hnfA (A:)
    gsmelrvgnryrlgrkigsgsfgdiylgtdiaageevaiklecvktkhpqlhieskiykm
    mqggvgiptirwcgaegdynvmvmellgpsledlfnfcsrkfslktvllladqmisriey
    ihsknfihrdvkpdnflmglgkkgnlvyiidfglakkyrdarthqhipyrenknltgtar
    yasinthlgieqsrrddleslgyvlmyfnlgslpwqglkaatkrqkyerisekkmstpie
    vlckgypsefatylnfcrslrfddkpdysylrqlfrnlfhrqgfsydyvfdwnmlk
    

    Sequence, based on observed residues (ATOM records): (download)
    >4hnfA (A:)
    lrvgnryrlgrkigsgsfgdiylgtdiaageevaiklecvkpqlhieskiykmmqggvgi
    ptirwcgaegdynvmvmellgpsledlfnfcsrkfslktvllladqmisrieyihsknfi
    hrdvkpdnflmglgkkgnlvyiidfglakkyrdarthqhipyrenknltgtaryasinth
    lgieqsrrddleslgyvlmyfnlgslpwqglkaatkrqkyerisekkmstpievlckgyp
    sefatylnfcrslrfddkpdysylrqlfrnlfhrqgfsydyvfdwnmlk
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >4hnfB (B:)
    gsmelrvgnryrlgrkigsgsfgdiylgtdiaageevaiklecvktkhpqlhieskiykm
    mqggvgiptirwcgaegdynvmvmellgpsledlfnfcsrkfslktvllladqmisriey
    ihsknfihrdvkpdnflmglgkkgnlvyiidfglakkyrdarthqhipyrenknltgtar
    yasinthlgieqsrrddleslgyvlmyfnlgslpwqglkaatkrqkyerisekkmstpie
    vlckgypsefatylnfcrslrfddkpdysylrqlfrnlfhrqgfsydyvfdwnmlk
    

    Sequence, based on observed residues (ATOM records): (download)
    >4hnfB (B:)
    vgnryrlgrkigsgsfgdiylgtdiaageevaiklecvktkhpqlhieskiykmmqggvg
    iptirwcgaegdynvmvmellgpsledlfnfcsrkfslktvllladqmisrieyihsknf
    ihrdvkpdnflmglgkkgnlvyiidfglakkyrdarthqhipyrenknltgtaryasint
    hlgieqsrrddleslgyvlmyfnlgslpwqglkaatkrqkyerisekkmstpievlckgy
    psefatylnfcrslrfddkpdysylrqlfrnlfhrqgfsydyvfdwnmlk