PDB entry 4hdf
View 4hdf on RCSB PDB site
Description: Crystal Structure of HIV-1 protease mutants V82A complexed with inhibitor GRL-0519
Class: HYDROLASE/Hydrolase Inhibitor
Keywords: aspartic acid protease, drug resistance, HIV-1 protease inhibitor GRL-0519, HYDROLASE-Hydrolase Inhibitor complex
Deposited on
2012-10-02, released
2013-08-14
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-08-14, with a file datestamp of
2013-08-09.
Experiment type: XRAY
Resolution: 1.29 Å
R-factor: 0.163
AEROSPACI score: 0.76
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: hiv-1 protease
Species: Human immunodeficiency virus type 1 [TaxId:11686]
Gene: gag-pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (32)
- engineered mutation (62)
- engineered mutation (66)
- engineered mutation (81)
- engineered mutation (94)
Domains in SCOPe 2.08: d4hdfa_ - Chain 'B':
Compound: hiv-1 protease
Species: Human immunodeficiency virus type 1 [TaxId:11686]
Gene: gag-pol
Database cross-references and differences (RAF-indexed):
- Uniprot P03367 (0-98)
- engineered mutation (6)
- engineered mutation (32)
- engineered mutation (62)
- engineered mutation (66)
- engineered mutation (81)
- engineered mutation (94)
Domains in SCOPe 2.08: d4hdfb_ - Heterogens: CL, G52, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>4hdfA (A:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
qiiieiaghkaigtvlvgptpaniigrnlltqigatlnf
- Chain 'B':
Sequence; same for both SEQRES and ATOM records: (download)
>4hdfB (B:)
pqitlwkrplvtikiggqlkealldtgaddtvieemslpgrwkpkmiggiggfikvrqyd
qiiieiaghkaigtvlvgptpaniigrnlltqigatlnf