PDB entry 4g2y
View 4g2y on RCSB PDB site
Description: Crystal structure of PDE5A complexed with its inhibitor
Class: hydrolase/hydrolase inhibitor
Keywords: phosphodiesterase, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2012-07-13, released
2013-06-26
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-06-26, with a file datestamp of
2013-06-21.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.183
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cGMP-specific 3',5'-cyclic phosphodiesterase
Species: Homo sapiens [TaxId:9606]
Gene: PDE5, PDE5A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4g2ya1, d4g2ya2 - Heterogens: PEG, ZN, MG, NI5, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4g2yA (A:)
mgsshhhhhhssglvprgshmeetrelqslaaavvpsaqtlkitdfsfsdfelsdletal
ctirmftdlnlvqnfqmkhevlcrwilsvkknyrknvayhnwrhafntaqcmfaalkagk
iqnkltdleilalliaalshdldhrgvnnsyiqrsehplaqlychsimehhhfdqclmil
nspgnqilsglsieeykttlkiikqailatdlalyikrrgeffelirknqfnledphqke
lflamlmtacdlsaitkpwpiqqriaelvateffdqgdrerkelnieptdlmnrekknki
psmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalaeqq
Sequence, based on observed residues (ATOM records): (download)
>4g2yA (A:)
meetrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhe
vlcrwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalsh
dldhrgvnnsplaqlychsimehhhfdqclmilnspgnqilsglsieeykttlkiikqai
latdlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpwpiqqriae
lvateffdknkipsmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalae