PDB entry 4f9y
View 4f9y on RCSB PDB site
Description: Human P38 alpha MAPK In Complex With a Novel and Selective Small Molecule Inhibitor
Class: transferase/transferase inhibitor
Keywords: protein kinase catalytic domain, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-05-21, released
2013-06-05
The last revision prior to the SCOPe 2.05 freeze date was dated
2013-07-24, with a file datestamp of
2013-07-19.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.169
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2, SAPK2A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4f9ya_ - Heterogens: GG5, LM3, BME, PEG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4f9yA (A:)
mhhhhhhssgvdlgtenlyfqsnasqerptfyrqelnktiwevperyqnlspvgsgaygs
vcaafdtktglrvavkklsrpfqsiihakrtyrelrllkhmkhenviglldvftparsle
efndvylvthlmgadlnnivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnla
vnedcelkildfglarhtddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaell
tgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiga
nplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqsfesrdllidew
ksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>4f9yA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglavatrwyrapeim
lnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkisses
arnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdp
ddepvadpydqsfesrdllidewksltydevisfvpppl