PDB entry 4f63
View 4f63 on RCSB PDB site
Description: Crystal structure of Human Fibroblast Growth Factor Receptor 1 Kinase domain in complex with compound 1
Class: transferase/transferase inhibitor
Keywords: kinase, ATP binding, phosphorylation, trans-membrane, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-05-14, released
2012-06-06
The last revision prior to the SCOPe 2.03 freeze date was dated
2012-06-27, with a file datestamp of
2012-06-22.
Experiment type: XRAY
Resolution: 2.55 Å
R-factor: 0.232
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4f63a_ - Chain 'B':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4f63b_ - Heterogens: 0S7, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4f63A (A:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>4f63A (A:)
elpedprwelprdrlvlgkplgqvvlaeaiglpnrvtkvavkmlksdatekdlsdlisem
emmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrppeeqlsskdlvsca
yqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihhidyykkttngrlpv
kwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelfkllkeghrmdkpsn
ctnelymmmrdcwhavpsqrptfkqlvedldrivalts
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4f63B (B:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>4f63B (B:)
seyelpedprwelprdrlvlgkplgegagqvvlaeaiglpnrvtkvavkmlksdatekdl
sdlisememmkmigkhkniinllgactqdgplyviveyaskgnlreylqarrqlsskdlv
scayqvargmeylaskkcihrdlaarnvlvtednvmkiadfgladyykkgrlpvkwmape
alfdriythqsdvwsfgvllweiftlggspypgvpveelfkllkeghrmdkpsnctnely
mmmrdcwhavpsqrptfkqlvedldrivalt