PDB entry 4eh8
View 4eh8 on RCSB PDB site
Description: Human p38 MAP kinase in complex with NP-F7 and RL87
Class: Transferase/Transferase inhibitor
Keywords: MAP Kinase Insert, Kinase-Ligand Complex, NP-Fragment, Transferase-Transferase inhibitor complex
Deposited on
2012-04-02, released
2012-12-05
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-01-02, with a file datestamp of
2012-12-28.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.242
AEROSPACI score: 0.33
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2, SAPK2A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4eh8a_ - Heterogens: IRG, 0OP, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4eh8A (A:)
gsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>4eh8A (A:)
erptfyrqelnktiwevperyqnlspvgsygsvcaafdtktglrvavkklsrpfqsiiha
krtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltdd
hvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfvatrwyrapeimlnwm
hynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarny
iqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddep
vadpydqsfesrdllidewksltydevisfvpppld