PDB entry 4dtk
View 4dtk on RCSB PDB site
Description: Novel and selective pan-PIM kinase inhibitor
Class: transferase/transferase inhibitor
Keywords: PIM1, Kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2012-02-21, released
2012-07-11
The last revision prior to the SCOPe 2.03 freeze date was dated
2012-07-25, with a file datestamp of
2012-07-20.
Experiment type: XRAY
Resolution: 1.86 Å
R-factor: 0.166
AEROSPACI score: 0.52
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase pim-1
Species: Homo sapiens [TaxId:9606]
Gene: PIM1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d4dtka_ - Heterogens: EDO, 7LI, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4dtkA (A:)
ekeplesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpme
vvllkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffw
qvleavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysp
pewiryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirw
clalrpsdrptfeeiqnhpwmqdvllpqetaeihlh
Sequence, based on observed residues (ATOM records): (download)
>4dtkA (A:)
plesqyqvgpllgsggfgsvysgirvsdnlpvaikhvekdrisdwgelpngtrvpmevvl
lkkvssgfsgvirlldwferpdsfvlilerpepvqdlfdfitergalqeelarsffwqvl
eavrhchncgvlhrdikdenilidlnrgelklidfgsgallkdtvytdfdgtrvysppew
iryhryhgrsaavwslgillydmvcgdipfehdeeiirgqvffrqrvssecqhlirwcla
lrpsdrptfeeiqnhpwmqdvllpqetaeihlh