PDB entry 4ctc
View 4ctc on RCSB PDB site
Description: Structure of the Human Anaplastic Lymphoma Kinase in Complex with the inhibitor 7-amino-3-cyclopropyl-12-fluoro-1,10,16-trimethyl-16,17- dihydro-1H-8,4-(metheno)pyrazolo(4,3-h)(2,5,11) benzoxadiazacyclotetradecin-15(10H)-one
Class: transferase
Keywords: transferase, inhibitor
Deposited on
2014-03-12, released
2014-05-28
The last revision prior to the SCOPe 2.06 freeze date was dated
2014-06-25, with a file datestamp of
2014-06-20.
Experiment type: XRAY
Resolution: 2.03 Å
R-factor: 0.1938
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: ALK tyrosine kinase receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4ctca_ - Heterogens: J99, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ctcA (A:)
mahhhhhhnpnycfagktssisdlkevprknitlirglghgafgevyegqvsgmpndpsp
lqvavktlpevcseqdeldflmealiiskfnhqnivrcigvslqslprfillelmaggdl
ksflretrprpsqpsslamldllhvardiacgcqyleenhfihrdiaarnclltcpgpgr
vakigdfgmardiyrasyyrkggcamlpvkwmppeafmegiftsktdtwsfgvllweifs
lgympypsksnqevlefvtsggrmdppkncpgpvyrimtqcwqhqpedrpnfaiilerie
yctqdpdvintalpieygplveeeekv
Sequence, based on observed residues (ATOM records): (download)
>4ctcA (A:)
pnycfagktssisdlkevprknitlirglggevyegqvplqvavktlpevcseqdeldfl
mealiiskfnhqnivrcigvslqslprfillelmaggdlksflretrprpsqpsslamld
llhvardiacgcqyleenhfihrdiaarnclltcpgpgrvakigdfgmardiggcamlpv
kwmppeafmegiftsktdtwsfgvllweifslgympypsksnqevlefvtsggrmdppkn
cpgpvyrimtqcwqhqpedrpnfaiilerieyctqdpdvintalpieyg