PDB entry 4btk

View 4btk on RCSB PDB site
Description: TTBK1 in complex with inhibitor
Class: transferase
Keywords: transferase, structure-kinetics relationship
Deposited on 2013-06-18, released 2013-09-25
The last revision prior to the SCOPe 2.06 freeze date was dated 2013-12-25, with a file datestamp of 2013-12-20.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.1922
AEROSPACI score: 0.37 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: tau-tubulin kinase 1
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d4btka_
  • Heterogens: DMS, DTQ, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4btkA (A:)
    mhhhhhhssgvdlgtenlyfqsnamqclaaalkdetnmsgggeqadilpanyvvkdrwkv
    lkkiggggfgeiyeamdlltrenvalkvesaqqpkqvlkmevavlkklqgkdhvcrfigc
    grnekfnyvvmqlqgrnladlrrsqprgtftlsttlrlgkqilesieaihsvgflhrdik
    psnfamgrlpstyrkcymldfglarqytnttgdvrpprnvagfrgtvryasvnahknrem
    grhddlwslfymlvefavgqlpwrkikdkeqvgmikekyehrmllkhmpsefhlfldhia
    sldyftkpdyqlimsvfensmkergiaeneafdweka
    

    Sequence, based on observed residues (ATOM records): (download)
    >4btkA (A:)
    dilpanyvvkdrwkvlkkigggeiyeamdlltrenvalkvesaqqpkqvlkmevavlkkl
    qgkdhvcrfigcgrnekfnyvvmqlqgrnladlrrsqprgtftlsttlrlgkqilesiea
    ihsvgflhrdikpsnfamgrlpstyrkcymldfglarqytnttgdvrpprnvagfrgtvr
    yasvnahknremgrhddlwslfymlvefavgqlpwrkikdkeqvgmikekyehrmllkhm
    psefhlfldhiasldyftkpdyqlimsvfensmkergiaeneafdwe