PDB entry 4a9u

View 4a9u on RCSB PDB site
Description: crystal structure of human chk2 in complex with benzimidazole carboxamide inhibitor
Class: transferase
Keywords: transferase
Deposited on 2011-11-28, released 2012-10-10
The last revision prior to the SCOPe 2.06 freeze date was dated 2012-11-07, with a file datestamp of 2012-11-02.
Experiment type: XRAY
Resolution: 2.48 Å
R-factor: 0.1854
AEROSPACI score: 0.37 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: serine/threonine-protein kinase chk2
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed):
    • Uniprot O96017 (7-End)
      • expression tag (6)
    Domains in SCOPe 2.06: d4a9ua1, d4a9ua2
  • Heterogens: NO3, EDO, A9U, CL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4a9uA (A:)
    gplgshmsvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsar
    eadpalnveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkea
    tcklyfyqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmr
    tlcgtptylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqits
    gkynfipevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllsee
    nestalpqvlaqpstsrkrpregeaegae
    

    Sequence, based on observed residues (ATOM records): (download)
    >4a9uA (A:)
    msvypkalrdeyimsktlgsevklaferktckkvaikiiskdpalnveteieilkklnhp
    ciikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengi
    ihrdlkpenvllssqeedclikitdfghskiltslmrtlcgtptylapevlvsvgtagyn
    ravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkk
    llvvdpkarftteealrhpwlqdedmkrkfqdllseenestalpqvla