PDB entry 3zr7

View 3zr7 on RCSB PDB site
Description: structural basis for agonism and antagonism for a set of chemically related progesterone receptor modulators
Class: receptor
Keywords: receptor, agonist, antagonist
Deposited on 2011-06-15, released 2011-08-17
The last revision prior to the SCOPe 2.06 freeze date was dated 2011-10-26, with a file datestamp of 2011-10-21.
Experiment type: XRAY
Resolution: 1.65 Å
R-factor: 0.16452
AEROSPACI score: 0.61 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: progesterone receptor
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d3zr7a_
  • Chain 'B':
    Compound: progesterone receptor
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.06: d3zr7b_
  • Heterogens: OR8, GOL, SO4, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >3zr7A (A:)
    gshmgqdiqlipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkws
    kslpgfrnlhiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkess
    fyslcltmwqipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyireli
    kaiglrqkgvvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmsevi
    aaqlpkilagmvkpllfhkk
    

    Sequence, based on observed residues (ATOM records): (download)
    >3zr7A (A:)
    lipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkwskslpgfrnl
    hiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkessfyslcltmw
    qipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyirelikaiglrqkg
    vvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmseviaaqlpkila
    gmvkpllfhk
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >3zr7B (B:)
    gshmgqdiqlipplinllmsiepdviyaghdntkpdtssslltslnqlgerqllsvvkws
    kslpgfrnlhiddqitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkess
    fyslcltmwqipqefvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyireli
    kaiglrqkgvvsssqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmsevi
    aaqlpkilagmvkpllfhkk
    

    Sequence, based on observed residues (ATOM records): (download)
    >3zr7B (B:)
    lipplinllmsiepdviyaghdntssslltslnqlgerqllsvvkwskslpgfrnlhidd
    qitliqyswmslmvfglgwrsykhvsgqmlyfapdlilneqrmkessfyslcltmwqipq
    efvklqvsqeeflcmkvllllntipleglrsqtqfeemrssyirelikaiglrqkgvvss
    sqrfyqltklldnlhdlvkqlhlyclntfiqsralsvefpemmseviaaqlpkilagmvk
    pllfhk