PDB entry 3wzk
View 3wzk on RCSB PDB site
Description: CRYSTAL STRUCTURE OF HUMAN MPS1 CATALYTIC DOMAIN IN COMPLEX WITH N-cyclopropyl-4-(8-((thiophen-2-ylmethyl)amino)imidazo[1,2-a]pyrazin-3-yl)benzamide
Class: transferase
Keywords: TRANSFERASE, ATP Binding, Phosphorylation
Deposited on
2014-09-29, released
2015-02-11
The last revision prior to the SCOPe 2.06 freeze date was dated
2015-02-11, with a file datestamp of
2015-02-06.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.224
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity protein kinase TTK
Species: Homo sapiens [TaxId:9606]
Gene: TTK, MPS1, MPS1L1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3wzka_ - Heterogens: CL, O23, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3wzkA (A:)
mecisvkgriysilkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiay
lnklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmlea
vhtihqhgivhsdlkpanflivdgmlklidfgianqmqpdttsvvkdsqvgtvnymppea
ikdmsssrengkskskispksdvwslgcilyymtygktpfqqiinqisklhaiidpnhei
efpdipekdlqdvlkcclkrdpkqrisipellahpyvqiqthpvnqmakgtteemkyvlg
qlvglnlvprgsaaghhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3wzkA (A:)
ecisvkgriysilkqigsggsskvfqvlnekkqiyaikyvnleeadnqtldsyrneiayl
nklqqhsdkiirlydyeitdqyiymvmecgnidlnswlkkkksidpwerksywknmleav
htihqhgivhsdlkpanflivdgmlklidfgianqmqpdgtvnymppeaikdmsispksd
vwslgcilyymtygktpfqqiinqisklhaiidpnheiefpdipekdlqdvlkcclkrdp
kqrisipellahpyvqiq