PDB entry 3uvr
View 3uvr on RCSB PDB site
Description: Human p38 MAP Kinase in Complex with KM064
Class: transferase/transferase inhibitor
Keywords: protein kinase, selective p38 inhibitor, SAR, annulen derivative, pyrazolo urea, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-11-30, released
2012-12-19
The last revision prior to the SCOPe 2.03 freeze date was dated
2012-12-19, with a file datestamp of
2012-12-14.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: 0.206
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3uvra_ - Heterogens: 06F, BOG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3uvrA (A:)
gsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3uvrA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglatrwyrapeimln
wmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesar
nyiqslkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepva
dpydqsfesrdllidewksltydevisfvpp