PDB entry 3u9n
View 3u9n on RCSB PDB site
Description: X-ray crystal structure of compound 1 bound to human CHK1 kinase domain
Class: transferase/transferase inhibitor
Keywords: Protein kinase domain, ATPase, ATP Binding, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-10-19, released
2012-01-25
The last revision prior to the SCOPe 2.06 freeze date was dated
2012-02-01, with a file datestamp of
2012-01-27.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: 0.197
AEROSPACI score: 0.46
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3u9na_ - Heterogens: 09H, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3u9nA (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgak
Sequence, based on observed residues (ATOM records): (download)
>3u9nA (A:)
edwdlvqtlgegaygevqlavnrvteeavavkivdenikkeicinkmlnhenvvkfyghr
regniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikpe
nlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvwsc
givltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsari
tipdikkdrwynkplkkg