PDB entry 3shy
View 3shy on RCSB PDB site
Description: Crystal structure of the PDE5A1 catalytic domain in complex with novel inhibitors
Class: hydrolase/hydrolase inhibitor
Keywords: PDE5A INHIBITOR, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-06-17, released
2011-08-24
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-11-08, with a file datestamp of
2017-11-03.
Experiment type: XRAY
Resolution: 2.65 Å
R-factor: N/A
AEROSPACI score: 0.18
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cGMP-specific 3',5'-cyclic phosphodiesterase
Species: Homo sapiens [TaxId:9606]
Gene: PDE5, PDE5A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3shya_ - Heterogens: 5FO, ZN, MG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3shyA (A:)
mgsshhhhhhssglvprgshmeetrelqslaaavvpsaqtlkitdfsfsdfelsdletal
ctirmftdlnlvqnfqmkhevlcrwilsvkknyrknvayhnwrhafntaqcmfaalkagk
iqnkltdleilalliaalshdldhrgvnnsyiqrsehplaqlychsimehhhfdqclmil
nspgnqilsglsieeykttlkiikqailatdlalyikrrgeffelirknqfnledphqke
lflamlmtacdlsaitkpwpiqqriaelvateffdqgdrerkelnieptdlmnrekknki
psmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalaeqq
Sequence, based on observed residues (ATOM records): (download)
>3shyA (A:)
etrelqslaaavvpsaqtlkitdfsfsdfelsdletalctirmftdlnlvqnfqmkhevl
crwilsvkknyrknvayhnwrhafntaqcmfaalkagkiqnkltdleilalliaalshdl
dhrgvnnsyiqrsehsimehhhfdqclmilnspgnqilsglsieeykttlkiikqailat
dlalyikrrgeffelirknqfnledphqkelflamlmtacdlsaitkpwpiqqriaelva
teffdqkknkipsmqvgfidaiclqlyealthvsedcfplldgcrknrqkwqalaeqq