PDB entry 3roc
View 3roc on RCSB PDB site
Description: Crystal structure of human p38 alpha complexed with a pyrimidinone compound
Class: Transferase/Transferase Inhibitor
Keywords: Transferase, Transferase-Transferase Inhibitor complex
Deposited on
2011-04-25, released
2011-06-15
The last revision prior to the SCOPe 2.03 freeze date was dated
2011-06-29, with a file datestamp of
2011-06-24.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.239
AEROSPACI score: 0.48
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2, THP-1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3roca_ - Heterogens: 29A, 29B, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3rocA (A:)
msqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3rocA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglvatrwyrapeiml
nwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesa
rnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpd
depvadpydqsfesrdllidewksltydevisfvppp