PDB entry 3qsd
View 3qsd on RCSB PDB site
Description: Structure of cathepsin B1 from Schistosoma mansoni in complex with CA074 inhibitor
Class: hydrolase/hydrolase inhibitor
Keywords: cysteine peptidase, digestive tract, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-02-21, released
2011-08-10
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-10-26, with a file datestamp of
2011-10-21.
Experiment type: XRAY
Resolution: 1.3 Å
R-factor: 0.116
AEROSPACI score: 0.8
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cathepsin B-like peptidase (C01 family)
Species: Schistosoma mansoni [TaxId:6183]
Gene: cb1.1, Smp_103610
Database cross-references and differences (RAF-indexed):
- Uniprot Q8MNY2 (Start-253)
- engineered mutation (98)
- engineered mutation (213)
Domains in SCOPe 2.06: d3qsda_ - Heterogens: 074, PEG, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qsdA (A:)
veipssfdsrkkwprcksiatirdqsrcgscwafgaveamsdrsciqsggkqnvelsavd
llsccescglgceggilgpawdywvkegivtgsskenhagcepypfpkcehhtkgkyppc
gskiyktprckqtcqkkyktpytqdkhrgkssynvkndekaiqkeimkygpveagftvye
dflnyksgiykhitgetlgghairiigwgvenkapywlianswnedwgengyfrivrgrd
ecsiesevtagrin
Sequence, based on observed residues (ATOM records): (download)
>3qsdA (A:)
eipssfdsrkkwprcksiatirdqsrcgscwafgaveamsdrsciqsggkqnvelsavdl
lsccescglgceggilgpawdywvkegivtgsskenhagcepypfpkcehhtkgkyppcg
skiyktprckqtcqkkyktpytqdkhrgkssynvkndekaiqkeimkygpveagftvyed
flnyksgiykhitgetlgghairiigwgvenkapywlianswnedwgengyfrivrgrde
csiesevtagrin