PDB entry 3qpp
View 3qpp on RCSB PDB site
Description: Structure of PDE10-inhibitor complex
Class: hydrolase/hydrolase inhibitor
Keywords: Phosphodiesterase Inhibitors, Structure-based drug design, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-02-14, released
2011-06-15
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-07-20, with a file datestamp of
2011-07-15.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.186
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: cAMP and cAMP-inhibited cGMP 3',5'-cyclic phosphodiesterase 10A
Species: Rattus norvegicus [TaxId:10116]
Gene: PDE10A
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3qppa_ - Heterogens: ZN, MG, SO4, DMS, PFW, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qppA (A:)
mhhhhhhssglvprgsamgtseewqglmhfnlparicrdielfhfdigpfenmwpgifvy
mihrscgtscfeleklcrfimsvkknyrrvpyhnwkhavtvahcmyailqnnnglftdle
rkglliaclchdldhrgfsnsylqkfdhplaalyststmeqhhfsqtvsilqleghnifs
tlssseyeqvleiirkaiiatdlalyfgnrkqleemyqtgslnlhnqshrdrviglmmta
cdlcsvtklwpvtkltandiyaefwaegdemkklgiqpipmmdrdkrdevpqgqlgfyna
vaipcyttltqilpptepllkacrdnlnqwekvirgeetamwisgpatskstsekptrkv
dd
Sequence, based on observed residues (ATOM records): (download)
>3qppA (A:)
nlparicrdielfhfdigpfenmwpgifvymihrscgtscfeleklcrfimsvkknyrrv
pyhnwkhavtvahcmyailqnnnglftdlerkglliaclchdldhrgfsnsylqkfdhpl
aalyststmeqhhfsqtvsilqleghnifstlssseyeqvleiirkaiiatdlalyfgnr
kqleemyqtgslnlhnqshrdrviglmmtacdlcsvtklwpvtkltandiyaefwaegde
mkklgiqpipmmdrdkrdevpqgqlgfynavaipcyttltqilpptepllkacrdnlnqw
ekvir