PDB entry 3qd4
View 3qd4 on RCSB PDB site
Description: Phosphoinositide-Dependent Kinase-1 (PDK1) kinase domain with 1,1-Dimethylethyl{(3R,5R)-1-[2-amino-6-(3-amino-1H-indazol-6-yl)-4-pyrimidinyl]-5-methyl-3-piperidinyl}carbamate
Class: transferase/transferase inhibitor
Keywords: kinase domain, AGC kinase, signal tranduction, ATP & Phosphoinositide, Phosphorylation on S241, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2011-01-17, released
2011-03-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-11-16, with a file datestamp of
2011-11-11.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: 0.199
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide-dependent protein kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: PDK1, PDPK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3qd4a_ - Heterogens: 3Q6, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qd4A (A:)
gpamdgtaaeprpgagslqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsre
yaikilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngel
lkyirkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgta
kvlspeskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragne
ylifqkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtw
enlhqqtppklt
Sequence, based on observed residues (ATOM records): (download)
>3qd4A (A:)
ppqprkkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtre
rdvmsrldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeiv
saleylhgkgiihrdlkpenillnedmhiqitdfgtakvlsgtaqyvspellteksacks
sdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvldat
krlgceemegygplkahpffesvtwenlhqqtppkl