PDB entry 3qci
View 3qci on RCSB PDB site
Description: Human receptor protein tyrosine phosphatase gamma, domain 1, in complex with N-[(3-aminophenyl)sulfonyl]-3-[(3,4-dichlorobenzyl)sulfanyl]thiophene-2-carboxamide
Class: hydrolase/hydrolase inhibitor
Keywords: TYROSINE RECEPTOR PHOSPHATASE, TWISTED MIXED BETA-SHEETS FLANKED BY {ALPHA}-HELICES, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2011-01-16, released
2011-12-28
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-12-28, with a file datestamp of
2011-12-23.
Experiment type: XRAY
Resolution: 2.27 Å
R-factor: 0.24
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Receptor-type tyrosine-protein phosphatase gamma
Species: Homo sapiens [TaxId:9606]
Gene: PTPG, PTPRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3qcia_ - Heterogens: NX3, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3qciA (A:)
gshmgsmeaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhkn
ryinilaydhsrvklrplpgkdskhsdyinanyvdgynkakayiatqgplkstfedfwrm
iweqntgiivmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirn
tkvkkgqkgnpkgrqnervviqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlv
hcsagvgrtgtyividsmlqqikdkstvnvlgflkhirtqrnylvqteeqyifihdalle
ailgketevs
Sequence, based on observed residues (ATOM records): (download)
>3qciA (A:)
meaipvkqfvkhigelysnnqhgfsedfeevqrctadmnitaehsnhpenkhknryinil
aydhsrvklrplpskhsdyinanyvdgynkakayiatqgplkstfedfwrmiweqntgii
vmitnlvekgrrkcdqywptenseeygniivtlkstkihacytvrrfsirntkvkqnerv
viqyhytqwpdmgvpeyalpvltfvrrssaarmpetgpvlvhcsagvgrtgtyividsml
qqikdkstvnvlgflkhirtqrnylvqteeqyifihdalleailg