PDB entry 3q6w
View 3q6w on RCSB PDB site
Description: Structure of dually-phosphorylated MET receptor kinase in complex with an MK-2461 analog with specificity for the activated receptor
Class: transferase/transferase inhibitor
Keywords: Tyrosine Kinase, two phosphotyrosine resiudes, transferase-transferase inhibitor complex
Deposited on
2011-01-03, released
2011-01-19
The last revision prior to the SCOPe 2.03 freeze date was dated
2011-06-22, with a file datestamp of
2011-06-17.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.205
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3q6wa_ - Heterogens: Q6W, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3q6wA (A:)
qntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihc
avkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrn
firnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglar
dmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdv
ntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfige
hhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3q6wA (A:)
tvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcav
kslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrnfi
rnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglardm
ydkeyysvhnklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdvntfdit
vyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfigehhhhh