PDB entry 3pg3
View 3pg3 on RCSB PDB site
Description: Human p38 MAP Kinase in Complex with RL182
Class: transferase/transferase inhibitor
Keywords: DFG-out, SAR, Kinase domain, Thiazole-urea, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-10-29, released
2011-11-02
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-11-02, with a file datestamp of
2011-10-28.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.221
AEROSPACI score: 0.41
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
- Uniprot Q16539
- engineered mutation (118)
- engineered mutation (161)
- engineered mutation (326)
Domains in SCOPe 2.02: d3pg3a_ - Heterogens: BOG, DG7, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pg3A (A:)
gsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivksq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglcrhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqslesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3pg3A (A:)
erptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsii
hakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivksqklt
ddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfgatrwyrapeimln
wmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesar
nyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpdd
epvadpydqslesrdllidewksltydevisfvpppl