PDB entry 3pe6
View 3pe6 on RCSB PDB site
Description: Crystal Structure of a soluble form of human MGLL in complex with an inhibitor
Class: hydrolase/hydrolase inhibitor
Keywords: alpha-beta hydrolase fold, Lipase, 2-arachidonyl-glycerol, Membrane associated, HYDROLASE, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2010-10-25, released
2011-03-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2013-06-19, with a file datestamp of
2013-06-14.
Experiment type: XRAY
Resolution: 1.35 Å
R-factor: 0.115
AEROSPACI score: 0.77
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Monoglyceride lipase
Species: Homo sapiens [TaxId:9606]
Gene: MGLL, hCG_40840
Database cross-references and differences (RAF-indexed):
- Uniprot Q6IBG9
- engineered mutation (35)
- engineered mutation (168)
- engineered mutation (175)
Domains in SCOPe 2.08: d3pe6a_ - Heterogens: ZYH, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3pe6A (A:)
mpeessprrtpqsipyqdlphlvnadgqylfcrywaptgtpkalifvshgagehsgryee
larmlmgldllvfahdhvghgqsegermvvsdfhvfvrdvlqhvdsmqkdypglpvfllg
hsmggaiailtaaerpghfagmvlisplvlanpesattfkvlaakvlnsvlpnlssgpid
ssvlsrnktevdiynsdplicraglkvcfgiqllnavsrveralpkltvpflllqgsadr
lcdskgayllmelaksqdktlkiyegayhvlhkelpevtnsvfheinmwvsqrtatagta
spp
Sequence, based on observed residues (ATOM records): (download)
>3pe6A (A:)
prrtpqsipyqdlphlvnadgqylfcrywaptgtpkalifvshgagehsgryeelarmlm
gldllvfahdhvghgqsegermvvsdfhvfvrdvlqhvdsmqkdypglpvfllghsmgga
iailtaaerpghfagmvlisplvlanpesattfkvlaakvlnsvlpnlssgpidssvlsr
nktevdiynsdplicraglkvcfgiqllnavsrveralpkltvpflllqgsadrlcdskg
ayllmelaksqdktlkiyegayhvlhkelpevtnsvfheinmwvsqrta