PDB entry 3p9j
View 3p9j on RCSB PDB site
Description: Aurora A kinase domain with phthalazinone pyrazole inhibitor
Class: transferase/transferase inhibitor
Keywords: Phosphotransferase, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-10-17, released
2011-03-23
The last revision prior to the SCOPe 2.03 freeze date was dated
2011-10-05, with a file datestamp of
2011-09-30.
Experiment type: XRAY
Resolution: 2.8 Å
R-factor: 0.204
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase 6
Species: Homo sapiens [TaxId:9606]
Gene: AIK, ARK1, AURA, AURKA, BTAK, STK15, STK6
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3p9ja_ - Heterogens: P9J, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3p9jA (A:)
akrqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreve
iqshlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelana
lsychskrvihrdikpenlllgsagelkiadfgwsvhapssrraalcgtldylppemieg
rmhdekvdlwslgvlcyeflvgkppfeantyqetykrisrveftfpdfvtegardlisrl
lkhnpsqrpmlrevlehpwitansskps
Sequence, based on observed residues (ATOM records): (download)
>3p9jA (A:)
rqwaledfeigrplgkgkfgnvylarekqskfilalkvlfkaqlekagvehqlrreveiq
shlrhpnilrlygyfhdatrvylileyaplgtvyrelqklskfdeqrtatyitelanals
ychskrvihrdikpenlllgsagelkiadfgwsvgtldylppemiegdekvdlwslgvlc
yeflvgkppfeantyqetykrisrveftfpdfvtegardlisrllkhnpsqrpmlrevle
hpwitanss