PDB entry 3ot8
View 3ot8 on RCSB PDB site
Description: X-ray crystal structure of compound 17r bound to human Chk1 kinase domain
Class: transferase/transferase inhibitor
Keywords: kinase, phosphatase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-09-10, released
2010-11-10
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-01-05, with a file datestamp of
2010-12-31.
Experiment type: XRAY
Resolution: 1.65 Å
R-factor: 0.179
AEROSPACI score: 0.55
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3ot8a_ - Heterogens: MI5, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3ot8A (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgak
Sequence, based on observed residues (ATOM records): (download)
>3ot8A (A:)
pfvedwdlvqtlgeggevqlavnrvteeavavkivdmnikkeicinkmlnhenvvkfygh
rrqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikpenll
lderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvwscgiv
ltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsaritip
dikkdrwynkplkkg