PDB entry 3new
View 3new on RCSB PDB site
Description: p38-alpha complexed with Compound 10
Class: transferase/transferase inhibitor
Keywords: Kinase, Ser/Thr kinase, Intracellular, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2010-06-09, released
2010-12-01
The last revision prior to the SCOPe 2.06 freeze date was dated
2011-03-30, with a file datestamp of
2011-03-25.
Experiment type: XRAY
Resolution: 2.51 Å
R-factor: 0.219
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2
Database cross-references and differences (RAF-indexed):
- Uniprot Q16539
- engineered mutation (167)
Domains in SCOPe 2.06: d3newa_ - Heterogens: 3NE
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3newA (A:)
gshmlemsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkk
lsrpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadln
nivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglarh
tddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlkl
ilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsd
kritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppld
qeemes
Sequence, based on observed residues (ATOM records): (download)
>3newA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcltddh
vqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglatrwyrapeimlnwm
hynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarny
iqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddep
vadpydqsfesrdllidewksltydevisfvppp