PDB entry 3nax
View 3nax on RCSB PDB site
Description: PDK1 in complex with inhibitor MP7
Class: transferase
Keywords: Kinase, Serine/threonine protein kinase, TRANSFERASE
Deposited on
2010-06-02, released
2010-11-24
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-04-06, with a file datestamp of
2011-04-01.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.166
AEROSPACI score: 0.56
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3-phosphoinositide-dependent protein kinase 1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3naxa_ - Heterogens: MP7, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3naxA (A:)
mhhhhhhenlyfqgqhaqpppqprkkrpedfkfgkilgegsfstvvlarelatsreyaik
ilekrhiikenkvpyvtrerdvmsrldhpffvklyftfqddeklyfglsyakngellkyi
rkigsfdetctrfytaeivsaleylhgkgiihrdlkpenillnedmhiqitdfgtakvls
peskqaransfvgtaqyvspellteksackssdlwalgciiyqlvaglppfragneylif
qkiikleydfpekffpkardlvekllvldatkrlgceemegygplkahpffesvtwenlh
qqtppkltayl
Sequence, based on observed residues (ATOM records): (download)
>3naxA (A:)
kkrpedfkfgkilgegsfstvvlarelatsreyaikilekrhiikenkvpyvtrerdvms
rldhpffvklyftfqddeklyfglsyakngellkyirkigsfdetctrfytaeivsaley
lhgkgiihrdlkpenillnedmhiqitdfgtakvlspeskqaraqyvspellteksacks
sdlwalgciiyqlvaglppfragneylifqkiikleydfpekffpkardlvekllvldat
krlgceemegygplkahpffesvtwenlhqqtppklta