PDB entry 3len
View 3len on RCSB PDB site
Description: Human Aldose Reductase mutant T113S complexed with Zopolrestat
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: Tim Barrel, T113S mutant, Oxidoreductase, NADP, Phosphoprotein, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2010-01-15, released
2011-01-19
The last revision prior to the SCOPe 2.08 freeze date was dated
2011-08-24, with a file datestamp of
2011-08-19.
Experiment type: XRAY
Resolution: 1.21 Å
R-factor: 0.124
AEROSPACI score: 0.86
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: aldose reductase
Species: Homo sapiens [TaxId:9606]
Gene: ALR2
Database cross-references and differences (RAF-indexed):
- Uniprot P15121 (Start-315)
- see remark 999 (4)
- engineered mutation (113)
Domains in SCOPe 2.08: d3lena_ - Heterogens: NAP, ZST, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3lenA (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwpsgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfheef
Sequence, based on observed residues (ATOM records): (download)
>3lenA (A:)
srillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiqek
lreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwpsgfkpgkef
fpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykpav
nqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaakhn
kttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvcall
sctshkdypfheef