PDB entry 3l8x
View 3l8x on RCSB PDB site
Description: P38 alpha kinase complexed with a pyrazolo-pyrimidine based inhibitor
Class: transferase
Keywords: p38 map kinase, serine/threonine-protine kinase, transferase
Deposited on
2010-01-04, released
2010-03-02
The last revision prior to the SCOPe 2.06 freeze date was dated
2010-03-02, with a file datestamp of
2010-02-26.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.225
AEROSPACI score: 0.28
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3l8xa_ - Heterogens: N4D, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3l8xA (A:)
mahhhhhsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkk
lsrpfqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadln
nivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarh
tddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlkl
ilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsd
kritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppld
qeemes
Sequence, based on observed residues (ATOM records): (download)
>3l8xA (A:)
erptfyrqelnktiwevperyqnlspvsvcaafdtktglrvavkklsrpfqsiihakrty
relrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkqkltddhvqfl
iyqilrglkyihsadiihrdlkpsnlavnedcelkildfglaratrwyrapeimnqtvdi
wsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsltqmp
kmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqs
fesrdllidewksltydevisfvppp