PDB entry 3kq7
View 3kq7 on RCSB PDB site
Description: Structure of human p38alpha with N-[4-methyl-3-(6-{[2-(1-methylpyrrolidin-2-yl)ethyl]amino}pyridine-3-amido)phenyl]-2-(morpholin-4-yl)pyridine-4-carboxamide
Class: transferase
Keywords: p38alpha kinase, alternative splicing, ATP binding, cytoplasm, kinase, nucleotide-binding, nucleus, phosphoprotein, polymorphism, serine/threonine-protein kinase, transferase
Deposited on
2009-11-17, released
2009-12-01
The last revision prior to the SCOPe 2.05 freeze date was dated
2009-12-01, with a file datestamp of
2009-11-27.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.19
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase p38 alpha
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d3kq7a_ - Heterogens: KQ7, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3kq7A (A:)
mgsshhhhhhssglvprgshmsqerptfyrqelnktiwevperyqnlspvgsgaygsvca
afdtktglrvavkklsrpfqsiihakrtyrelrllkhmkhenviglldvftparsleefn
dvylvthlmgadlnnivkcqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavne
dcelkildfglarhtddemtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgr
tlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqsltqmpkmnfanvfiganpl
avdllekmlvldsdkritaaqalahayfaqyhdpddepvadpydqsfesrdllidewksl
tydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3kq7A (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemtgyva
trwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpga
ellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqala
hayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvppp