PDB entry 3k3i
View 3k3i on RCSB PDB site
Description: p38alpha bound to novel DGF-out compound PF-00215955
Class: transferase
Keywords: P38 Kinase, Alternative splicing, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase
Deposited on
2009-10-02, released
2009-11-17
The last revision prior to the SCOPe 2.03 freeze date was dated
2009-12-08, with a file datestamp of
2009-12-04.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.196
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2, P38
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.03: d3k3ia_ - Heterogens: JZJ, I46, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3k3iA (A:)
gsrptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsi
ihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkl
tddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemtgy
vatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtp
gaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqa
lahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvppp
Sequence, based on observed residues (ATOM records): (download)
>3k3iA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnikltddhvq
fliyqilrglkyihsadiihrdlkpsnlavnedcelkildfgvatrwyrapeimlnwmhy
nqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiq
sltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepva
dpydqsfesrdllidewksltydevisfvppp