PDB entry 3iw8
View 3iw8 on RCSB PDB site
Description: Structure of Inactive Human p38 MAP Kinase in Complex with a Thiazole-Urea
Class: transferase
Keywords: DFG-out, Type-III, Thiazole, Alternative splicing, ATP-binding, Cytoplasm, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase
Deposited on
2009-09-02, released
2009-11-17
The last revision prior to the SCOPe 2.05 freeze date was dated
2010-01-05, with a file datestamp of
2009-12-31.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.22
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
- Uniprot Q16539
- engineered (118)
- engineered (161)
- engineered (326)
Domains in SCOPe 2.05: d3iw8a_ - Heterogens: HIZ, BOG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3iw8A (A:)
gsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivksq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglcrhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqslesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>3iw8A (A:)
erptfyrqelnktiwevperyqnlspvgsygsvcaafdtktglrvavkklsrpfqsiiha
krtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivksqkltdd
hvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfgatrwyrapeimlnwm
hynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarny
iqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddep
vadpydqslesrdllidewksltydevisfvppp