PDB entry 3i5n
View 3i5n on RCSB PDB site
Description: Crystal structure of c-Met with triazolopyridazine inhibitor 13
Class: transferase
Keywords: proto-oncogene, RTK, receptor tyrosine kinase, scatter factor receptor, HGF/SF, Alternative splicing, ATP-binding, Chromosomal rearrangement, Disease mutation, Disulfide bond, Glycoprotein, Kinase, Membrane, Nucleotide-binding, Phosphoprotein, Polymorphism, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2009-07-06, released
2010-01-12
The last revision prior to the SCOPe 2.02 freeze date was dated
2010-01-12, with a file datestamp of
2010-01-08.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.225
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3i5na_ - Heterogens: B2D, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3i5nA (A:)
qntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihc
avkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlrn
firnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglar
dmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdv
ntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfige
hyvhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3i5nA (A:)
hidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkihcavks
lnrevsqfltegiimkdfshpnvlsllgiclplvvlpymkhgdlrnfirnethnptvkdl
igfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfglardmydkeyysvhklp
vkwmaleslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpe
ycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig