PDB entry 3hec
View 3hec on RCSB PDB site
Description: P38 in complex with Imatinib
Class: transferase
Keywords: Transferase, ATP-binding, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Serine/threonine-protein kinase
Deposited on
2009-05-08, released
2009-11-10
The last revision prior to the SCOPe 2.02 freeze date was dated
2010-08-18, with a file datestamp of
2010-08-13.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.222
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: CSBP, CSBP1, CSBP2, CSPB1, MAPK14, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.02: d3heca_ - Heterogens: STI, BOG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3hecA (A:)
rptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrpfqsiih
akrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltd
dhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtddemtgyva
trwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpga
ellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkritaaqala
hayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvppp
Sequence, based on observed residues (ATOM records): (download)
>3hecA (A:)
rptfyrqelnktiwevperyqnlspvgsvcaafdtktglrvavkklsrpfqsiihakrty
relrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltddhvqf
liyqilrglkyihsadiihrdlkpsnlavnedcelkildfatrwyrapeimlnwmhynqt
vdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqslt
qmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpy
dqsfesrdllidewksltydevisfvppp