PDB entry 3h8c
View 3h8c on RCSB PDB site
Description: A combined crystallographic and molecular dynamics study of cathepsin-L retro-binding inhibitors (compound 14)
Class: hydrolase
Keywords: Cysteine Proteases, Cathepsin L, Disulfide bond, Glycoprotein, Hydrolase, Lysosome, Protease, Thiol protease, Zymogen
Deposited on
2009-04-29, released
2009-10-20
The last revision prior to the SCOPe 2.06 freeze date was dated
2014-11-12, with a file datestamp of
2014-11-07.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.237
AEROSPACI score: 0.21
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cathepsin L1
Species: Homo sapiens [TaxId:9606]
Gene: Cathepsin L
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3h8ca_ - Chain 'B':
Compound: Cathepsin L1
Species: Homo sapiens [TaxId:9606]
Gene: Cathepsin L
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3h8cb_ - Heterogens: NSZ, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3h8cA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestesdnn
kywlvknswgeewgmggyvkmakdrrnhcgiasaasyptv
Sequence, based on observed residues (ATOM records): (download)
>3h8cA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfesnkywlv
knswgeewgmggyvkmakdrrnhcgiasaasyptv
- Chain 'B':
Sequence, based on SEQRES records: (download)
>3h8cB (B:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestesdnn
kywlvknswgeewgmggyvkmakdrrnhcgiasaasyptv
Sequence, based on observed residues (ATOM records): (download)
>3h8cB (B:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfesnkywlv
knswgeewgmggyvkmakdrrnhcgiasaasyptv