PDB entry 3gxj
View 3gxj on RCSB PDB site
Description: Structure of Alk5 + GW855857
Class: transferase
Keywords: TGF-beta, Alk5, kinase, inhibitor, quinazoline, Aortic aneurysm, ATP-binding, Craniosynostosis, Disease mutation, Disulfide bond, Glycoprotein, Magnesium, Manganese, Membrane, Metal-binding, Nucleotide-binding, Phosphoprotein, Polymorphism, Receptor, Serine/threonine-protein kinase, Transferase, Transmembrane
Deposited on
2009-04-02, released
2009-04-21
The last revision prior to the SCOPe 2.08 freeze date was dated
2009-06-23, with a file datestamp of
2009-06-19.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.223
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d3gxja_ - Heterogens: 855, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3gxjA (A:)
iartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhenil
gfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhmei
vgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkryma
pevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsvee
mrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqqeg
ikm
Sequence, based on observed residues (ATOM records): (download)
>3gxjA (A:)
iartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhenil
gfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhmei
vgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiagtkrymapevld
dsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsveemrkvv
ceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqq